indium in-111

Small moleculeapproved

Approved

Dec 29, 1992

Indium In-111 pentetate disodium is a radioactive diagnostic indicated for use in radionuclide cisternography. Decay of In-111 by electron capture allows for detection with a gamma camera for visualization of the brain and spinal column. Indium In 111 pentetate ( 111In-DTPA) is indicated as an imaging agent in cisternography to study the flow of cerebrospinal fluid (CSF) in the brain, to diagnose abnormalities in CSF circulation, to assess and help localize the site of CSF leakage, and to test the patency of or localize blocks in CSF shunts. — NCATS

Clinical trial activity

1 trials · 2 clinical orgs · 2 marketing orgs

Phase 1
0
Phase 2
0
Phase 3
0
Phase 4
0

Earliest trial started Jul 1, 2007 (NCT00602862)

Timeline

1990s

  1. Dec 29, 1992

    General Electric — Earliest FDA Approval

  2. Dec 29, 1992

    General Electric — NDA Secondary Org

  3. Dec 29, 1992

    General Electric — NDA Organization

  4. Sep 27, 1994

    Curium Pharma — NDA Secondary Org

Indications

Mechanism of action

  • Unspecified targetOTHER

    Diagnostic agent

  • contrast mediumRadiopaque

    contrast medium radiopaque

Approval history

  • approvedDec 29, 1992

Chemistry & pharmacology

Loading structure…

SMILES

[111In+3]
Mol. weight
221.18 g/mol
Chirality
Achiral Molecule
Inorganic
Yes
Polymer
No
Delivery
Parenteral
Availability
Discontinued

Oral

No

Parenteral

Yes

Topical

No

Sources

Also known as

  • 111in-bevacizumab
  • (111)indium chloride
  • 111indium trichloride
  • 111indium trichloride
  • (113)indium chloride
  • indiclor
  • indiclor
  • indiclor
  • indium
  • indium
  • indium-111 chloride
  • indium-111 chloride
  • indium (111in) chloride injection
  • indium chloride
  • indium chloride
  • indium chloride
  • indium chloride (111incl3)
  • indium chloride (111incl3)
  • indium chloride in-111
  • indium chloride in-111
  • indium chloride (incl3)
  • indium in-111
  • indium in 111 chloride
  • indium in 111 chloride
  • indium in 111 chloride
  • indium in-111 chloride
  • indium in-111 chloride
  • indium in-111 chloride
  • indium in-111 chloride solution
  • indium in 111m chloride
  • indium in 111m chloride
  • indium in-111m chloride
  • indium in-111m chloride
  • indium trichloride
  • indium trichloride, 111in-labeled
  • indium trichloride (113)
  • indium trichloride, 113in-labeled

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT00602862N/AJul 1, 2007Dutch Cancer Society, Radboud University
Showing 1 of 1 trials
Page 1 / 1

Organizations

Research & Development (2)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
Dutch Cancer SocietyAcademic/Hospital1012007
Radboud UniversityAcademic/Hospital1112007
2 organizations
Page 1 / 1

Marketing (3)

OrganizationOrg typeRelationshipDate
Curium PharmaFor profitNDA2Sep 27, 1994
General ElectricFor profitNDA2Dec 29, 1992
General ElectricFor profitNDADec 29, 1992