fadrozole monohydrochloride
Small moleculeexperimental
Clinical trial activity
0 trials · 0 clinical orgs · 0 marketing orgs
Phase 1
0
Phase 2
0
Phase 3
0
Phase 4
0
Mechanism of action
- Cytochrome P450 19A1INHIBITOR
Cytochrome P450 19A1 inhibitor
Can bind to CYP11B1 and B2 (different enantiomers of fadrozole bind each enzyme).
Chemistry & pharmacology
Loading structure…
SMILES
N#Cc1ccc(C2CCCc3cncn32)cc1- Mol. weight
- 223.28 g/mol
- Lipinski Ro5
- Pass
- Rule of 3
- Yes
- Chirality
- Racemic Mixture
- Inorganic
- No
- Polymer
- No
Oral
No
Parenteral
No
Topical
No
Sources
- ChEMBLCHEMBL9298 ↗
- ChEMBLCHEMBL468419 ↗
Also known as
- cgs 16949a
- cgs-16949a
- fadrozole
- fadrozole
- fadrozole
- fadrozole
- fadrozole
- fadrozole
- fadrozole hcl
- fadrozole hydrochloride
- fadrozole monohydrochloride