ethoheptazine
Small moleculeexperimental
Ethoheptazine is an analgesic, which belongs to the proheptazine group. It was used either alone (Zactane trade name) or in combination with meprobamate and aspirin (Equagesic) for the pain relief in patients with headache or musculoskeletal disorders. Currently all mediactions containing ethoheptazine are withdrawn from the market. The exact target of ethoheptazine is unknow, but it is believed that it may have modulatory effect on opioid receptors. — NCATS
Clinical trial activity
0 trials · 0 clinical orgs · 0 marketing orgs
Phase 1
0
Phase 2
0
Phase 3
0
Phase 4
0
Indications
Approved for
Chemistry & pharmacology
Loading structure…
SMILES
CCOC(=O)C1(c2ccccc2)CCCN(C)CC1- Mol. weight
- 261.36 g/mol
- Lipinski Ro5
- Pass
- Rule of 3
- Yes
- Chirality
- Racemic Mixture
- Inorganic
- No
- Polymer
- No
Oral
No
Parenteral
No
Topical
No
Sources
- ChEMBLCHEMBL170797 ↗
- WikipediaEthoheptazine ↗
- NCATS3A4G3A848U ↗
- ChEMBLCHEMBL1201887 ↗
Also known as
- aethoheptazin
- ethoheptazine
- ethoheptazine
- ethoheptazine
- ethoheptazine citrate
- ethoheptazine citrate
- ethoheptazine citrate
- ethoheptazine citrate
- ethoheptazine citrate
- ethyl heptazine