amisometradine

Small moleculeexperimental

AMISOMETRADINE, a pyrimidinedione-based diuretic, is an isomer of aminometradine with less toxicity and a reasonable diuretic potency. — NCATS

Clinical trial activity

0 trials · 0 clinical orgs · 0 marketing orgs

Phase 1
0
Phase 2
0
Phase 3
0
Phase 4
0

Chemistry & pharmacology

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SMILES

CN1C(=O)C=C(N)N(CC(C)=C)C1=O
Mol. weight
195.2184 g/mol
Lipinski Ro5
Pass
Rule of 3
No
Chirality
Achiral Molecule
Inorganic
No
Polymer
No

Oral

No

Parenteral

No

Topical

No

Sources

Also known as

  • aminoisometradin
  • aminoisometradine
  • amisometradin
  • amisometradine
  • amisometradine
  • amisometradine
  • amisometradine