stryphnone
Small moleculeexperimental
Adrenalone is a keton form of the natural substrate epinephrine. Adrenalone is evidently formed in vivo by hydrolytic cleavage of the diester by esterases. It is an adrenergic receptor agonist. Adrenalone inhibits the norepinephrine synthesis and dopamine beta oxidase. It is known to have very weak sympathomimetic activity when compared to adrenaline. Adrenalone has the high radioprotective effect. It is a topical nasal decongestant. Adrenalone has hemostatic, sympathomimetic and vasoconstrictor therapeutic functions. — NCATS
Clinical trial activity
0 trials · 0 clinical orgs · 0 marketing orgs
Phase 1
0
Phase 2
0
Phase 3
0
Phase 4
0
Indications
Approved for
Chemistry & pharmacology
Loading structure…
SMILES
CNCC(=O)C1=CC=C(O)C(O)=C1- Mol. weight
- 181.1885 g/mol
- Lipinski Ro5
- Pass
- Rule of 3
- No
- Chirality
- Achiral Molecule
- Inorganic
- No
- Polymer
- No
Oral
No
Parenteral
No
Topical
No
Sources
- NCATSEGU41QL329 ↗
- ChEMBLCHEMBL2103996 ↗
Also known as
- 4-methylaminoacetopyrocatechol
- adrenalone
- adrenalone
- adrenalone
- adrenalone
- adrenalone
- adrenon
- adrenone
- methaminoacetocatech
- stryphnon
- stryphnone