octanoic acid

Small moleculeexperimental

OCTANOIC ACID (Caprylic acid) eight-carbon saturated fatty acid belongs to the class of mediumchain saturated fatty acids. OCTANOIC ACID found naturally in the milk of various mammals, and as a minor constituent of coconut oil and palm kernel oil. Caprylic acid is used commercially in the production of esters used in perfumery and also in the manufacture of dyes. Caprylic acid is an antimicrobial pesticide used as a food contact surface sanitizer in commercial food handling establishments on dairy equipment, food processing equipment, breweries, wineries, and beverage processing plants. It is also used as disinfectant in health care facilities, schools/colleges, animal care/veterinary facilities, industrial facilities, office buildings, recreational facilities, retail and wholesale establishments, livestock premises, restaurants, and hotels/motels. In addition, caprylic acid is used as an algaecide, bactericide, and fungicide in nurseries, greenhouses, garden centers, and interiorscapes on ornamentals. Products containing caprylic acid are formulated as soluble concentrate/liquids and ready-to-use liquids. — NCATS

Clinical trial activity

9 trials · 15 clinical orgs · 0 marketing orgs

Phase 1
4
Phase 2
6
Phase 3
0
Phase 4
0

Earliest trial started Oct 1, 2004 (NCT00142805)

Timeline

2000s

  1. Jan 1, 2004

    Earliest Phase 2 Sponsor(trial)

  2. Jan 1, 2009

    Earliest Phase 1 Sponsor(trial)

Indications

Mechanism of action

  • Unspecified targetUnclear

    unclear

Chemistry & pharmacology

Loading structure…

SMILES

CCCCCCCC(O)=O
Mol. weight
144.2114 g/mol
Lipinski Ro5
Pass
Rule of 3
No
Chirality
Achiral Molecule
Inorganic
No
Polymer
No

Oral

No

Parenteral

No

Topical

No

Sources

Also known as

  • caprylic acid
  • caprylic acid
  • caprylic acid
  • caprylic acid
  • caprylic acid
  • caprylic acid, 14c-labeled
  • caprylic acid, aluminum salt
  • caprylic acid, ammonia salt
  • caprylic acid, barium salt
  • caprylic acid, cadmium salt
  • caprylic acid, calcium salt
  • caprylic acid, cesium salt
  • caprylic acid, chromium(+2) salt
  • caprylic acid, cobalt salt
  • caprylic acid, copper(+2) salt
  • caprylic acid, copper salt
  • caprylic acid, iridum(+3) salt
  • caprylic acid, iron(+3) salt
  • caprylic acid, lanthanum(+3) salt
  • caprylic acid, lead(+2) salt
  • caprylic acid, lithium salt
  • caprylic acid, manganese salt
  • caprylic acid, nickel(+2) salt
  • caprylic acid, potassium salt
  • caprylic acid, ruthenium(+3) salt
  • caprylic acid, sodium salt
  • caprylic acid, sodium salt, 11c-labeled
  • caprylic acid, tin(+2) salt
  • caprylic acid, tin salt
  • caprylic acid, zinc salt
  • caprylic acid, zirconium(+4) salt
  • caprylic acid, zirconium salt
  • capryloate
  • capryloate
  • caprylsaeure
  • caprylsaeure
  • n-octanoic acid
  • n-octanoic acid
  • n-octoic acid
  • n-octoic acid
  • n-octylic acid
  • n-octylic acid
  • octanoate
  • octanoate
  • octanoate
  • octanoic acid
  • octanoic acid
  • octanoic acid
  • octanoic acid
  • octanoic acid
  • octanoic acid
  • octanoic acid
  • octanoic acid
  • octic acid
  • octic acid
  • octoic acid
  • octoic acid
  • octylic acid
  • octylic acid
  • sodium caprate
  • sodium caprylate
  • sodium caprylate
  • sodium caprylate
  • sodium octanoate
  • sodium octanoate

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT02602158Early Phase 1 (Phase 1)Oct 1, 2015University of Zurich
NCT01864525Phase 1/Phase 2 (Phase 2)Jul 1, 2013National Institute on Deafness and Other Communication Disorders (NIDCD), Syracuse University
NCT03467737N/ADec 1, 2012Baylor University, Purdue University
NCT01433016Phase 2Nov 1, 2011Exalenz Bioscience LTD., Hebrew University, Henry Ford Health System, Medical University of South Carolina, Northwestern University, University of Toronto
NCT01468948Phase 1Oct 28, 2011National Institute of Neurological Disorders and Stroke (NINDS)
NCT01244503Phase 2Feb 1, 2011Exalenz Bioscience LTD., Virginia Commonwealth University
NCT00848172Phase 1/Phase 2 (Phase 2)Feb 1, 2009National Institute of Neurological Disorders and Stroke (NINDS)
NCT00355550Phase 2Jul 1, 2006Cerecin, Psychologix, Inc.
NCT00142805Phase 2Oct 1, 2004Cerecin
Showing 9 of 9 trials
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Organizations

Research & Development (15)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
CerecinFor profit2212004
Exalenz Bioscience LTD.For profit2112011
National Institute of Neurological Disorders and Stroke (NINDS)Government2222009
Baylor UniversityAcademic/Hospital1012012
Hebrew UniversityAcademic/Hospital1012011
Henry Ford Health SystemAcademic/Hospital1012011
Medical University of South CarolinaAcademic/Hospital1012011
National Institute on Deafness and Other Communication Disorders (NIDCD)Government1012013
Northwestern UniversityAcademic/Hospital1012011
Psychologix, Inc.For profit1012006
Purdue UniversityAcademic/Hospital1112012
Syracuse UniversityAcademic/Hospital1112013
University of TorontoAcademic/Hospital1012011
University of ZurichAcademic/Hospital1112015
Virginia Commonwealth UniversityAcademic/Hospital1112011
15 organizations
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