Laronidase

Trade name: Aldurazyme

Recombinant proteinapprovedOrphan Drug FDA

Approved

Apr 30, 2003

Iduronidase, sold as Aldurazyme, is an enzyme with the systematic name glycosaminoglycan α-L-iduronohydrolase. It catalyses the hydrolysis of unsulfated α-L-iduronosidic linkages in dermatan sulfate. — Wikipedia

Clinical trial activity

20 trials · 18 clinical orgs · 1 marketing orgs

Phase 1
8
Phase 2
9
Phase 3
4
Phase 4
4

Earliest trial started Dec 1, 2000 (NCT00912925)

Timeline

1990s

  1. Sep 24, 1997

    Orphan Drug Designation

2000s

  1. Jan 1, 2000

    Earliest Phase 3 Sponsor(trial)

  2. Jan 1, 2002

    Earliest Phase 2 Sponsor(trial)

  3. Apr 30, 2003

    Biomarin — Earliest FDA Approval

  4. Apr 30, 2003

    Biomarin — NDA Organization

  5. Apr 30, 2003

    Biomarin — Marketing Organization

  6. Jan 1, 2005

    Earliest Phase 1 Sponsor(trial)

Indications

Mechanism of action

Approval history

  • approvedApr 30, 2003

Chemistry & pharmacology

Chirality
Single Stereoisomer
Inorganic
No
Polymer
No
Delivery
Parenteral
Availability
Prescription Only
Multi-specific
No

Oral

No

Parenteral

Yes

Topical

No

Black box warning

Sources

Also known as

  • aldurazyme
  • aldurazyme
  • aldurazyme
  • aldurazyme
  • a-l-iduronidase
  • alpha-l-iduronidase
  • alpha-l-iduronidase precursor
  • human alpha iduronidase
  • laronidase
  • laronidase
  • laronidase
  • laronidase
  • laronidase
  • laronidase
  • laronidase
  • laronidase
  • laronidase
  • laronidase (genetical recombination)
  • ovine hyaluronidase
  • sperm adhesion molecule 1
  • sperm surface protein ph-20
  • vitrase
  • wydase
  • wydase
  • wydase

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT06406153Phase 3Sep 10, 2022Cinnagen
NCT05134571Phase 4Oct 28, 2021Genzyme, Sanofi
NCT04453085Phase 1/Phase 2 (Phase 2)May 1, 2021JCR Pharmaceuticals Co., Ltd.
NCT04532047Phase 1Dec 1, 2020Duke University, University of California, San Francisco
NCT04227600Phase 1/Phase 2 (Phase 2)Sep 1, 2020JCR Pharmaceuticals Co., Ltd.
NCT02232477N/AMay 1, 2014Los Angeles Biomedical Research Institute, National Institute of Neurological Disorders and Stroke (NINDS), National Institutes of Health (NIH), The Ryan Foundation, UCLA Medical Center, University of California, Los Angeles, University of California, San Francisco, University of Minnesota
NCT01173016Phase 1May 1, 2012University of Minnesota
NCT00418821Phase 4Oct 1, 2010Genzyme
NCT00852358N/AJun 1, 2009Biomarin, National Center for Advancing Translational Science (NCATS), National Institute of Diabetes and Digestive and Kidney Diseases (NIDDK), National Institute of Neurological Disorders and Stroke (NINDS), National Institutes of Health (NIH), The Ryan Foundation, University of California, Los Angeles, University of Minnesota, Washington University in St. Louis
NCT00741338Phase 1/Phase 2 (Phase 2)Sep 1, 2008Genzyme
NCT00638547Phase 1Jan 2, 2008University of Minnesota
NCT00786968Phase 1Jan 1, 2008The Ryan Foundation, University of California, Los Angeles, Washington University in St. Louis
NCT00258011Phase 3Dec 1, 2005Genzyme
NCT00215527Phase 1Nov 1, 2005Food and Drug Administration, The Ryan Foundation, University of California, Los Angeles, Washington University in St. Louis
NCT00144781Phase 4Dec 1, 2004Genzyme
NCT00144768Phase 4Jul 1, 2004Genzyme
NCT00176891Phase 2Mar 1, 2004University of Minnesota
NCT00146757Phase 2Oct 1, 2002Genzyme
NCT00146770Phase 3May 1, 2001Genzyme
NCT00912925Phase 3Dec 1, 2000Genzyme
Showing 20 of 20 trials
Page 1 / 1

Organizations

Research & Development (18)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
GenzymeFor profit9932000
University of MinnesotaAcademic/Hospital5332004
The Ryan FoundationAcademic/Hospital4022005
University of California, Los AngelesAcademic/Hospital4022005
Washington University in St. LouisAcademic/Hospital3322005
JCR Pharmaceuticals Co., Ltd.For profit2212020
National Institute of Neurological Disorders and Stroke (NINDS)Government2012009
National Institutes of Health (NIH)Government2012009
University of California, San FranciscoAcademic/Hospital2122014
BiomarinFor profit1012009
CinnagenFor profit1112022
Duke UniversityAcademic/Hospital1012020
Food and Drug AdministrationGovernment1012005
Los Angeles Biomedical Research InstituteAcademic/Hospital1012014
National Center for Advancing Translational Science (NCATS)Government1012009
National Institute of Diabetes and Digestive and Kidney Diseases (NIDDK)Government1012009
SanofiFor profit1012021
UCLA Medical CenterAcademic/Hospital1112014
18 organizations
Page 1 / 1

Marketing (2)

OrganizationOrg typeRelationshipDate
BiomarinFor profitNDAApr 30, 2003
BiomarinFor profitMKTGApr 30, 2003