am-461
Small moleculeexperimental
Clinical trial activity
0 trials · 0 clinical orgs · 0 marketing orgs
Phase 1
0
Phase 2
0
Phase 3
0
Phase 4
0
Mechanism of action
- G protein-coupled receptor 44ANTAGONIST
PTGDR2 antagonist
Indication: Allergic diseases
Chemistry & pharmacology
Loading structure…
SMILES
COc1ccc(CC(=O)O)cc1Oc1ccc(NC(=O)C(C)(C)C)cc1CSC(C)(C)C- Mol. weight
- 459.61 g/mol
- Lipinski Ro5
- 1 violation(s)
- Rule of 3
- No
- Chirality
- Single Stereoisomer
- Inorganic
- No
- Polymer
- No
Oral
No
Parenteral
No
Topical
No
Sources
- ChEMBLCHEMBL5095021 ↗
- ChEMBLCHEMBL3545014 ↗
Also known as
- am-461
- am-461