lodoxamide tromethamine

Trade name: alomide

Small moleculeapprovedOrphan Drug FDA

Approved

Sep 23, 1993

Lodoxamide is an antiallergic pharmaceutical drug. It is marketed under the tradename Alomide in the UK. Like cromoglicic acid it acts as a mast cell stabilizer. In 2014 lodoxamide and bufrolin were found to be potent agonists at the G protein-coupled receptor 35, an orphan receptor believed to play a role in inflammatory processes, pain and the development of stomach cancer. — Wikipedia

Clinical trial activity

0 trials · 0 clinical orgs · 1 marketing orgs

Phase 1
0
Phase 2
0
Phase 3
0
Phase 4
0

Timeline

1990s

  1. Oct 16, 1991

    Orphan Drug Designation

  2. Sep 23, 1993

    Novartis — Earliest FDA Approval

  3. Sep 23, 1993

    Novartis — NDA Organization

  4. Sep 23, 1993

    Novartis — NDA Secondary Org

Indications

Mechanism of action

Approval history

  • approvedSep 23, 1993

Chemistry & pharmacology

Loading structure…

SMILES

N#Cc1cc(NC(=O)C(=O)O)c(Cl)c(NC(=O)C(=O)O)c1.NC(CO)(CO)CO
Mol. weight
432.77 g/mol
Lipinski Ro5
Pass
Rule of 3
No
Inorganic
No
Polymer
No

Oral

No

Parenteral

No

Topical

No

Sources

Also known as

  • 2,2'-((2-chloro-5-cyano-1,3-phenylene)diimino)bis(2-oxoacetic acid), compd. with 2-amino-2- (hydroxymethyl)-1,3-propanediol (1:2)
  • alomide
  • alomide
  • alomide
  • alomide
  • alomide
  • alomide allergy
  • lodoxamide trometamol
  • lodoxamide trometamol
  • lodoxamide trometamol
  • lodoxamide tromethamine
  • lodoxamide tromethamine
  • lodoxamide tromethamine
  • lodoxamide tromethamine
  • lodoxamide tromethamine
  • lodoxamide tromethamine
  • u 42585 e
  • u-42585e
  • u-42585e
  • u-42,585e
  • u-42,585e

Organizations

Marketing (2)

OrganizationOrg typeRelationshipDate
NovartisFor profitNDASep 23, 1993
NovartisFor profitNDA2Sep 23, 1993