piperocaine monohydrochloride

Small moleculeexperimental

Piperocaine (Metycaine) is a local anesthetic drug. It is an ester and primarily is a sodium channel blocker. Piperocaine can partially inhibit dopamine. It is known as a alpha-1-proteinase inhibitor. Used in the form of its hydrochloride as a local or spinal anesthetic and in dental anesthesia. Can cause toxic reactions. Piperocaine Hydrochloride is in the list of Bulk Drug Substances Nominated for Use in Compounding Under Section 503A, FDA Act. Piperocaine hydrochloride is a small, white odorless crystals or a white crystalline powder, stable in air, freely soluble in water, alcohol and chloroform. — NCATS

Clinical trial activity

0 trials · 0 clinical orgs · 0 marketing orgs

Phase 1
0
Phase 2
0
Phase 3
0
Phase 4
0

Indications

Approved for

Chemistry & pharmacology

Loading structure…

SMILES

CC1CCCCN1CCCOC(=O)C2=CC=CC=C2
Mol. weight
261.3593 g/mol
Lipinski Ro5
Pass
Rule of 3
No
Chirality
Racemic Mixture
Inorganic
No
Polymer
No

Oral

No

Parenteral

No

Topical

No

Sources

Also known as

  • (+/-)-2-methyl-1-piperidinepropanol benzoate (ester)
  • 2-methylpiperidinepropanol benzoate
  • neothesin
  • piperocaine
  • piperocaine hydrochloride
  • piperocaine hydrochloride
  • piperocaine hydrochloride
  • piperocaine, (+-)-isomer
  • piperocaine monohydrochloride
  • piperocaine monohydrochloride, (+-)-isomer