methylphenobarbital

Small moleculeexperimental

Mephobarbital us a barbiturate derivative used primary as an anticonvulsant, but also as a sedative and anxiolytic. Marketing of mephobarbital was discontinued in 2012. — NCATS

Clinical trial activity

0 trials · 0 clinical orgs · 0 marketing orgs

Phase 1
0
Phase 2
0
Phase 3
0
Phase 4
0

Indications

Approved for

Chemistry & pharmacology

Loading structure…

SMILES

CCC1(C(=O)NC(=O)N(C)C1=O)C2=CC=CC=C2
Mol. weight
246.2619 g/mol
Lipinski Ro5
Pass
Rule of 3
No
Chirality
Racemic Mixture
Inorganic
No
Polymer
No

Oral

No

Parenteral

No

Topical

No

Sources

Also known as

  • 1-methylphenobarbital
  • 1-methylphenobarbital
  • 5-ethyl-1-methyl-5-phenyl-2,4,6(1h,3h,5h)-pyrimidinetrione
  • 5-ethyl-1-methyl-5-phenyl-2,4,6(1h,3h,5h)-pyrimidinetrione
  • 5-ethyl-1-methyl-5-phenylbarbituric acid
  • 5-ethyl-1-methyl-5-phenylbarbituric acid
  • 5-ethyl-1-methyl-5-phenyl-pyrimidine-2,4,6-trione
  • 5-ethyl-1-methyl-5-phenyl-pyrimidine-2,4,6-trione
  • enphenemal
  • enphenemal
  • enphenemal
  • mebaral
  • mebaral
  • menta-bal
  • menta-bal
  • mephobarbital
  • mephobarbital
  • mephobarbital
  • mephobarbital
  • mephobarbital
  • mephobarbital
  • mephobarbital
  • mephobarbitone
  • mephobarbitone
  • mephobarbitone
  • methylphenobarbital
  • methylphenobarbital
  • methylphenobarbital
  • methylphenobarbital
  • methylphenobarbital
  • methylphenobarbital
  • méthylphénobarbital
  • méthylphénobarbital
  • methylphenobarbitalum
  • methylphenobarbitalum
  • methylphenobarbitone
  • methylphenobarbitone
  • methylphenobarbitone
  • methylphenobarbitone
  • metilfenobarbital
  • metilfenobarbital
  • metilfenobarbitale
  • metilfenobarbitale
  • metylfenemal
  • n-methylphenobarbital
  • n-methylphenobarbital
  • prominal
  • prominal