octinoxate

Small moleculeapproved

Approved

Dec 7, 1992

Octinoxate, also called Octyl methoxycinnamate or (OMC), is a UV filter. It can be absorbed rapidly through skin.Octinoxate filters UV‐B rays from the sun, although it does not protect against UV-A rays. Octinoxate dissolves in oil, which makes it a fat-seeking substance in the body. It is formed by combining methoxycinnamic acid and 2-ethylhexanol compounds which are not harmful on their own. When mixed together, they form a clear liquid that does not dissolve in water. Octinoxate is found in hair color products and shampoos, sunscreen, lipstick, nail polish, and skin creams. In products other than sunscreens, it is used as a UV filter to protect the products from degrading when exposed to the sun. — NCATS

Clinical trial activity

2 trials · 2 clinical orgs · 1 marketing orgs

Phase 1
0
Phase 2
0
Phase 3
0
Phase 4
1

Earliest trial started Jul 1, 2008 (NCT00530387)

Timeline

1990s

  1. Dec 7, 1992

    Bayer — Earliest FDA Approval

  2. Dec 7, 1992

    Bayer — NDA Secondary Org

  3. Dec 7, 1992

    Bayer — NDA Organization

Indications

Mechanism of action

  • Unspecified targetUltraviolet filter

    ultraviolet filter

Combination products

Approval history

  • approvedDec 7, 1992

Chemistry & pharmacology

Loading structure…

SMILES

CCCCC(CC)COC(=O)C=Cc1ccc(OC)cc1
Mol. weight
290.4 g/mol
Lipinski Ro5
Pass
Rule of 3
No
Chirality
Racemic Mixture
Inorganic
No
Polymer
No
Delivery
Topical
Availability
Discontinued

Oral

No

Parenteral

No

Topical

Yes

Sources

Also known as

  • 2-ethylhexyl 3-(methoxyphenyl)-2-propenoate
  • 2-ethylhexyl-4-methoxycinnamate
  • 2-ethylhexyl-p-methoxycinnamate
  • ehmc cpd
  • escalol 557
  • ethylhexyl methoxycinnamate
  • ethylhexyl methoxycinnamate
  • ethylhexyl methoxycinnamate
  • ethylhexyl methoxycinnamate
  • ethylhexyl p-methoxycinnamate
  • ethylhexyl p-methoxycinnamate
  • ethylhexyl p-methoxycinnamate
  • eusolex 2292
  • heliopan new
  • methoxycinnamate
  • octinoxate
  • octinoxate
  • octinoxate
  • octinoxate
  • octinoxate
  • octinoxate
  • octinoxate
  • octinoxate
  • octylmethoxycinnamate
  • octyl methoxycinnamate
  • octyl methoxycinnamate
  • octyl methoxycinnamate
  • octyl methoxycinnamate
  • octyl methoxycinnamate
  • octyl methoxycinnamate
  • octyl-methoxycinnamate
  • omc cinnamate
  • parsol
  • parsol
  • parsol
  • parsol
  • parsol mcx
  • parsol mox
  • uvinul mc80

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT01695356Phase 4Sep 1, 2012Universidad Autonoma de San Luis Potosi
NCT00530387N/AJul 1, 2008University of Dundee
Showing 2 of 2 trials
Page 1 / 1

Organizations

Research & Development (2)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
Universidad Autonoma de San Luis PotosiAcademic/Hospital1112012
University of DundeeAcademic/Hospital1112008
2 organizations
Page 1 / 1

Marketing (2)

OrganizationOrg typeRelationshipDate
BayerFor profitNDA2Dec 7, 1992
BayerFor profitNDADec 7, 1992